Aspadol 100 mg Ingredients: Everything You Need to Know

Aspadol 100 mg is a prescription rapid pain relief medicine widely used to treat moderate to severe pain. It contains Tapentadol 100 mg as its main active ingredient, which makes it a powerful opioid analgesic. This article explains the composition of Aspadol 100 mg, its active and inactive ingredients, how these ingredients work, and why it is important to know what’s inside the medicine you take.

1. What is Aspadol 100 mg?

Aspadol 100mg is a pain-relieving opioids drugs that belongs to the class of centrally acting opioid analgesics. Doctors prescribe it when standard painkillers like paracetamol or NSAIDs (ibuprofen, diclofenac) are not sufficient. It is commonly used to manage pain caused by:

Post-surgical procedures
Injuries or trauma
Chronic back pain
Neuropathic pain (pain caused by nerve damage)
Joint and muscle pain, including rheumatoid arthritis and osteoarthritis

Aspadol Tablet Uses

Chronic pain management – Effective for long-term pain such as arthritis, lower back pain, and nerve pain.
Post-surgical pain – Helps control acute pain after surgery or major injury.
Musculoskeletal pain – Useful in conditions like sprains, strains, or orthopedic injuries.
Neuropathic pain – Provides relief in nerve-related pain that may not respond to regular painkillers.

Aspadol works via a dual mechanism: it acts on μ-opioid receptors to block pain signals and inhibits norepinephrine reuptake to enhance pain control.

2. Active Ingredient of Aspadol 100 mg

The main active ingredient of Aspadol 100mg is Tapentadol 100 mg.

What is Tapentadol?

Tapentadol is a centrally acting synthetic opioids painkiller that combines two mechanisms of action in one molecule:
1. Opioid receptor agonist – It binds to μ-opioid receptors in the brain and spinal cord to block pain signals.
2. Norepinephrine reuptake inhibitor – It increases norepinephrine levels, enhancing the body’s natural ability to control pain.

Why is Tapentadol used in Aspadol?

Strong pain relief: Works when mild painkillers fail.
Dual-action: Effective for both tissue pain (nociceptive pain) and nerve pain (neuropathic pain).
Rapid onset: Starts working quickly to provide fast pain control.
Better tolerability: Causes fewer gastrointestinal issues (like nausea and constipation) than some traditional opioids.

3. Inactive Ingredients of Aspadol 100 mg

Along with Tapentadol, Aspadol tablets contain pharmaceutical excipients (inactive substances). These ingredients do not treat pain but help the tablet maintain its shape, stability, and absorption in the body.

Common inactive ingredients include:

Microcrystalline cellulose – Used as a binder to hold the tablet together.
Povidone – Helps dissolve the medicine evenly in the stomach.
Magnesium stearate – Prevents sticking during tablet manufacturing.
Lactose monohydrate – Used as a filler (not suitable for lactose-intolerant patients).
Colloidal silicon dioxide – Improves tablet flow during production.
Film coating agents – Give the tablet a smooth finish and protect it from moisture.

Note: The exact excipient list may vary slightly depending on the manufacturer, but these are commonly used.

4. How the Ingredients Work Together

Tapentadol tablets (active salt) directly provides pain relief.
Excipients ensure that the drug is released properly, absorbed efficiently, and remains stable until use.
Film coating helps the tablet pass through the digestive tract without breaking down too early.

This combination ensures consistent pain control and a predictable effect, which is important for a medicine used to manage strong pain.

5. Why Knowing the Ingredients is Important

Understanding the ingredients of Aspadol 100mg is useful for several reasons:

Allergy awareness: Some patients may be allergic to certain excipients like lactose or povidone.
Drug safety: Knowing the active salt helps prevent accidental overdose if you are taking other Tapentadol-based medicines.
Interaction check: If you’re taking other opioids or sedatives, being aware of the active ingredient helps avoid harmful drug interactions.
Informed decisions: Patients who are cautious about opioid medicines can discuss alternatives with their doctor.

6. Dosage and Administration (Quick Note)

The usual adult dose for extended-release tablets is 100 mg every 12 hours, as prescribed by a doctor.
Swallow whole with water. Do not crush or chew the tablet to avoid rapid release of Tapentadol.
Do not exceed the prescribed dose to prevent risk of dependence, overdose, or breathing problems.

7. Safety Advice Related to Ingredients

Lactose intolerance: If you are lactose intolerant, check with your doctor about the excipients used.
Avoid alcohol and sedatives: Since Tapentadol is an opioid, mixing it with alcohol or sleeping pills can be dangerous.
Pregnancy and breastfeeding: Only use Aspadol tab if clearly prescribed by a doctor.
Liver or kidney disease: Patients with impaired organ function may need dosage adjustments.
Allergic reactions: If you notice rash, swelling, or breathing issues after taking the medicine, seek medical help immediately.

8. Key Takeaways About Aspadol 100 mg Ingredients

Active ingredient: Tapentadol 100 mg (powerful opioid painkiller).
Inactive ingredients: Excipients like microcrystalline cellulose, povidone, magnesium stearate, and lactose.
Purpose of ingredients: Active salt provides pain relief, while excipients ensure stability and proper absorption.
Patient awareness: Knowing what’s inside the tablet helps in identifying allergies, avoiding overdoses, and ensuring safe use.

Aspadol Variants (Strengths and Forms)

Aspadol is a brand name for Tapentadol, an opioid analgesic used to treat moderate to severe pain. It is available in different strengths and formulations to suit varying patient needs and pain severities. Below are the common Aspadol variants:

Aspadol 100 mg
Aspadol 50mg
Aspadol 75mg

9. Frequently Asked Questions (FAQs)

Q1. What is the active salt in Aspadol 100 mg?
The active salt is Tapentadol 100 mg, an opioid analgesic.

Q2. Can lactose-intolerant patients take Aspadol 100 mg?
Some formulations contain lactose as an excipient. Always check with your doctor or pharmacist before use.

Q3. Are there any herbal or food interactions with Aspadol ingredients?
Avoid alcohol, sedatives, and certain herbal products that cause drowsiness, as they can increase side effects.

Q4. Do inactive ingredients affect the pain relief of Aspadol?
No, inactive ingredients don’t treat pain. They are used to make the tablet stable, safe, and easy to swallow.

Q5. Can I take other opioid medicines with Aspadol 100 mg?
No, combining opioids increases the risk of overdose and breathing problems. Use only as prescribed.

Q6. Where can I buy Aspadol 100mg online?
You can purchase Aspadol 100 mg from trusted online pharmacies that sell genuine medicines. Always choose verified platforms like GenericsMedicineShop to ensure product authenticity, secure payments, and fast shipping.